Triptorelin initially causes a temporary increase in serum testosterone levels. Because of this, symptoms of prostate cancer may worsen during the first weeks of treatment. Notify your doctor if you experience new or worsening symptoms such as bone pain; blood in the urine; difficulty urinating; or numbness, tingling, weakness, or paralysis.
Triptorelin reduces the amount of testosterone produced in the body.
Triptorelin is used in the palliative treatment of advanced prostate cancer.
Triptorelin may also be used for purposes other than those listed in this medication guide.
Before using triptorelin, tell your doctor if you have
metastatic back bone (spinal) lesions, or
You may not be able to use triptorelin, or you may require a dosage adjustment or special monitoring during treatment.
Triptorelin is in the FDA pregnancy category X. This means that triptorelin will cause birth defects in an unborn baby.Triptorelin must be administered under the supervision of a physician.
Triptorelin is injected into the muscle, usually once a month.
Your doctor or nurse will rotate the site of the injection periodically.
Triptorelin initially causes a temporary increase in serum testosterone levels. Because of this, symptoms of prostate cancer may worsen during the first weeks of treatment. Notify your doctor if you experience new or worsening symptoms such as bone pain; blood in the urine; difficulty urinating; or numbness, tingling, weakness, or paralysis.
Triptorelin vials for injection should be stored at room temperature away from moisture and heat.
Contact your doctor if you miss a dose of triptorelin.
An overdose of triptorelin is unlikely to occur. If you do suspect that an overdose has occurred, contact your doctor, hospital emergency room, or poison control center for advice.
There are no restrictions on food, beverages, or activities while using triptorelin. Follow any special instructions given by your doctor.
an allergic reaction (difficulty breathing; closing of your throat; swelling of your lips, tongue, or face; or hives);
difficulty urinating or blood in the urine;
bone pain; or
numbness, tingling, weakness, or paralysis.
Other, less serious side effects may be more likely to occur. Talk to your doctor if you experience
increased blood pressure;
impotence;
nausea or vomiting;
dizziness;
headache; or
pain at the injection site.
Side effects other than those listed here may also occur. Talk to your doctor about any side effect that seems unusual or that is especially bothersome.
It is not known whether triptorelin will interact with other medicines. Talk to your doctor and pharmacist before taking any prescription or over-the-counter medicines, including herbal products during treatment with triptorelin.
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